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Yaser A. Mostafa
Yaser A. Mostafa
Associate Professor of Pharmaceutical Organic Chemistry, Assiut University
Verified email at pharm.aun.edu.eg
Title
Cited by
Cited by
Year
Thiohydantoin derivatives incorporating a pyrazole core: Design, synthesis and biological evaluation as dual inhibitors of topoisomerase-I and cycloxygenase-2 with anti-cancer …
KRA Abdellatif, WAA Fadaly, YA Mostafa, DM Zaher, HA Omar
Bioorganic Chemistry 91, 103132, 2019
432019
Synthesis and antimicrobial activity of certain new 1, 2, 4-triazolo [1, 5-a] pyrimidine derivatives
YAH Mostafa, MA Hussein, AA Radwan, AEHN Kfafy
Archives of pharmacal research 31, 279-293, 2008
412008
Steroid derivatives as inhibitors of steroid sulfatase
YAM Abdel-Karem
Journal of Steroid Biochemistry & Molecular Biology 137, 183– 198, 2013
40*2013
Inhibition of steroid sulfatase with 4-substituted estrone and estradiol derivatives
CM Phan, Y Liu, B Kim, Y Mostafa, SD Taylor
Bioorganic & medicinal chemistry 19 (20), 5999-6005, 2011
372011
Antioxidant and Wound Healing Potential of Vitis vinifera Seeds Supported by Phytochemical Characterization and Docking Studies
T Al-Warhi, EM Zahran, S Selim, MM Al-Sanea, MM Ghoneim, SA Maher, ...
Antioxidants 11 (5), 881, 2022
272022
Discovery of new pyrimido [5, 4-c] quinolines as potential antiproliferative agents with multitarget actions: Rapid synthesis, docking, and ADME studies
RA Mekheimer, SMR Allam, MA Al-Sheikh, MS Moustafa, SM Al-Mousawi, ...
Bioorganic Chemistry 121, 105693, 2022
272022
17β-Arylsulfonamides of 17β-aminoestra-1, 3, 5 (10)-trien-3-ol as highly potent inhibitors of steroid sulfatase
YA Mostafa, SD Taylor
Bioorganic & medicinal chemistry 20 (4), 1535-1544, 2012
242012
A first-in-class anticancer dual HDAC2/FAK inhibitors bearing hydroxamates/benzamides capped by pyridinyl-1, 2, 4-triazoles
M Mustafa, AA Abd El-Hafeez, D Abdelhamid, GD Katkar, YA Mostafa, ...
European journal of medicinal chemistry 222, 113569, 2021
212021
A facile synthesis, drug-likeness, and in silico molecular docking of certain new azidosulfonamide–chalcones and their in vitro antimicrobial activity
M Mustafa, YA Mostafa
Monatshefte für Chemie-Chemical Monthly 151, 417-427, 2020
192020
Wound Healing and Antioxidant Capabilities of Zizyphus mauritiana Fruits: In-Vitro, In-Vivo, and Molecular Modeling Study
NH Shady, R Soltane, SA Maher, EA Saber, MA Elrehany, YA Mostafa, ...
Plants 11 (11), 1392, 2022
162022
Novel urea linked ciprofloxacin-chalcone hybrids having antiproliferative topoisomerases I/II inhibitory activities and caspases-mediated apoptosis
HHH Mohammed, SH Abbas, AM Hayallah, GEDA Abuo-Rahma, ...
Bioorganic Chemistry 106, 104422, 2021
162021
Antimicrobial pyridazines: synthesis, characterization, cytotoxicity, substrate promiscuity, and molecular docking
M Mustafa, YA Mostafa
Chemistry & Biodiversity 17 (6), e2000100, 2020
162020
Novel piperine-carboximidamide hybrids: Design, synthesis, and antiproliferative activity via a multi-targeted inhibitory pathway
LH Al-Wahaibi, MA Mahmoud, YA Mostafa, AE Raslan, BGM Youssif
Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 376-386, 2023
152023
Synthesis and biological evaluation of indole-2-carboxamides with potent apoptotic antiproliferative activity as egfr/cdk2 dual inhibitors
LH Al-Wahaibi, YA Mostafa, MH Abdelrahman, AH El-Bahrawy, ...
Pharmaceuticals 15 (8), 1006, 2022
142022
A-ring substituted 17β-arylsulfonamides of 17β-aminoestra-1, 3, 5 (10)-trien-3-ol as highly potent reversible inhibitors of steroid sulfatase
YA Mostafa, B Kralt, PPN Rao, SD Taylor
Bioorganic & Medicinal Chemistry 23 (17), 5681-5692, 2015
132015
FAK inhibitors as promising anticancer targets: present and future directions
M Mustafa, AA Abd El-Hafeez, DA Abdelhafeez, D Abdelhamid, ...
Future Medicinal Chemistry 13 (18), 1559-1590, 2021
122021
Novel 1, 5-diaryl pyrazole-3-carboxamides as selective COX-2/sEH inhibitors with analgesic, anti-inflammatory, and lower cardiotoxicity effects
OM Hendawy, HAM Gomaa, SI Alzarea, MS Alshammari, FAM Mohamed, ...
Bioorganic Chemistry 116, 105302, 2021
112021
Discovery of new cyanopyridine/chalcone hybrids as dual inhibitors of EGFR/BRAFV600E with promising antiproliferative properties
HA Abou‐Zied, EAM Beshr, HAM Gomaa, YA Mostafa, BGM Youssif, ...
Archiv der Pharmazie 356 (4), 2200464, 2023
102023
Discovery of novel oxazole-based macrocycles as anti-coronaviral agents targeting SARS-CoV-2 main protease
LH Al-Wahaibi, A Mostafa, YA Mostafa, OF Abou-Ghadir, AH Abdelazeem, ...
Bioorganic Chemistry 116, 105363, 2021
102021
Novel indazole derivatives as potent apoptotic antiproliferative agents by multi-targeted mechanism: Synthesis and biological evaluation
FOA Frejat, H Zhai, Y Cao, L Wang, YA Mostafa, HAM Gomaa, ...
Bioorganic Chemistry 126, 105922, 2022
82022
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