| Designing focused chemical libraries enriched in protein-protein interaction inhibitors using machine-learning methods C Reynès, H Host, AC Camproux, G Laconde, F Leroux, A Mazars, ... PLoS computational biology 6 (3), e1000695, 2010 | 144 | 2010 |
| iPPI-DB: a manually curated and interactive database of small non-peptide inhibitors of protein–protein interactions CM Labbé, G Laconde, MA Kuenemann, BO Villoutreix, O Sperandio Drug discovery today 18 (19-20), 958-968, 2013 | 116 | 2013 |
| N-Acyl Benzotriazole Derivatives for the Synthesis of Dipeptides and Tripeptides and Peptide Biotinylation by Mechanochemistry L Gonnet, T Tintillier, N Venturini, L Konnert, JF Hernandez, F Lamaty, ... ACS Sustainable Chemistry & Engineering 5 (4), 2936-2941, 2017 | 90 | 2017 |
| A leap into the chemical space of protein-protein interaction inhibitors B O Villoutreix, C M Labbe, D Lagorce, G Laconde, O Sperandio Current pharmaceutical design 18 (30), 4648-4667, 2012 | 84 | 2012 |
| Drug to genome to drug: discovery of new antiplasmodial compounds TB Beghyn, J Charton, F Leroux, G Laconde, A Bourin, P Cos, L Maes, ... Journal of medicinal chemistry 54 (9), 3222-3240, 2011 | 64 | 2011 |
| Synthesis of five-and six-membered lactams via solvent-free microwave Ugi reaction M Jida, S Malaquin, R Deprez-Poulain, G Laconde, B Deprez Tetrahedron Letters 51 (39), 5109-5111, 2010 | 55 | 2010 |
| Design, synthesis and biological evaluation of substituted dioxodibenzothiazepines and dibenzocycloheptanes as farnesyltransferase inhibitors P Gilleron, N Wlodarczyk, R Houssin, A Farce, G Laconde, JF Goossens, ... Bioorganic & medicinal chemistry letters 17 (19), 5465-5471, 2007 | 53 | 2007 |
| Ugi reaction for the synthesis of 4-aminopiperidine-4-carboxylic acid derivatives. Application to the synthesis of carfentanil and remifentanil S Malaquin, M Jida, JC Gesquiere, R Deprez-Poulain, B Deprez, ... Tetrahedron Letters 51 (22), 2983-2985, 2010 | 50 | 2010 |
| Sol–gel synthesis of collagen-inspired peptide hydrogel C Echalier, S Jebors, G Laconde, L Brunel, P Verdié, L Causse, A Bethry, ... Materials Today 20 (2), 59-66, 2017 | 44 | 2017 |
| A dipteran’s novel sucker punch: Evolution of arthropod atypical venom with a neurotoxic component in robber flies (Asilidae, Diptera) SH Drukewitz, N Fuhrmann, EAB Undheim, A Blanke, J Giribaldi, R Mary, ... Toxins 10 (1), 29, 2018 | 41 | 2018 |
| Solvent-free microwave-assisted Meyers’ lactamization M Jida, R Deprez-Poulain, S Malaquin, P Roussel, ... Green Chemistry 12 (6), 961-964, 2010 | 39 | 2010 |
| Racemic and diastereoselective construction of indole alkaloids under solvent-and catalyst-free microwave-assisted Pictet–Spengler condensation M Jida, OM Soueidan, B Deprez, G Laconde, R Deprez-Poulain Green Chemistry 14 (4), 909-911, 2012 | 35 | 2012 |
| A facile and rapid synthesis of N-benzyl-2-substituted piperazines M Jida, M Soueidan, N Willand, F Agbossou-Niedercorn, L Pelinski, ... Tetrahedron letters 52 (14), 1705-1708, 2011 | 33 | 2011 |
| Tyrosine Kinase Syk Non-Enzymatic Inhibitors and Potential Anti-Allergic Drug-Like Compounds Discovered by Virtual and In Vitro Screening BO Villoutreix, G Laconde, D Lagorce, P Martineau, MA Miteva, ... PLoS One 6 (6), e21117, 2011 | 29 | 2011 |
| Water-based conditions for the microscale parallel synthesis of bicyclic lactams S Malaquin, M Jida, J Courtin, G Laconde, N Willand, B Deprez, ... Tetrahedron Letters 54 (6), 562-567, 2013 | 22 | 2013 |
| Stapled peptide targeting the CDK4/Cyclin D interface combined with Abemaciclib inhibits KRAS mutant lung cancer growth C Bouclier, M Simon, G Laconde, M Pellerano, S Diot, S Lantuejoul, ... Theranostics 10 (5), 2008, 2020 | 21 | 2020 |
| Synthesis, Structure and Biological Activity of CIA and CIB, Two α-Conotoxins from the Predation-Evoked Venom of Conus catus J Giribaldi, D Wilson, A Nicke, Y El Hamdaoui, G Laconde, A Faucherre, ... Toxins 10 (6), 222, 2018 | 17 | 2018 |
| Derivatives of Iressa, a specific epidermal growth factor receptor inhibitor, are powerful apoptosis inducers in PC3 prostatic cancer cells A Telliez, M Desroses, N Pommery, O Briand, A Farce, G Laconde, ... ChemMedChem: Chemistry Enabling Drug Discovery 2 (3), 318-332, 2007 | 16 | 2007 |
| New antiproliferative benzoindolinothiazepines derivatives G Laconde, P Depreux, P Berthelot, N Pommery, JP Hénichart European journal of medicinal chemistry 40 (2), 167-172, 2005 | 16 | 2005 |
| Synthesis of α-Amino Acid N-Carboxyanhydrides G Laconde, M Amblard, J Martinez Organic Letters 23 (16), 6412-6416, 2021 | 13 | 2021 |
