Back to the future: Advances in development of broad-spectrum capsid-binding inhibitors of enteroviruses A Egorova, S Ekins, M Schmidtke, V Makarov European journal of medicinal chemistry 178, 606-622, 2019 | 41 | 2019 |
Novel pleconaril derivatives: Influence of substituents in the isoxazole and phenyl rings on the antiviral activity against enteroviruses A Egorova, E Kazakova, B Jahn, S Ekins, V Makarov, M Schmidtke European journal of medicinal chemistry 188, 112007, 2020 | 37 | 2020 |
Pipeline of anti‐Mycobacterium abscessus small molecules: Repurposable drugs and promising novel chemical entities A Egorova, M Jackson, V Gavrilyuk, V Makarov Medicinal research reviews 41 (4), 2350-2387, 2021 | 35 | 2021 |
Small Molecules—Prospective Novel HCMV Inhibitors E Bogner, A Egorova, V Makarov Viruses 13 (3), 474, 2021 | 14 | 2021 |
Dispirotripiperazine-core compounds, their biological activity with a focus on broad antiviral property, and perspectives in drug design (mini-review) A Egorova, E Bogner, E Novoselova, KM Zorn, S Ekins, V Makarov European Journal of Medicinal Chemistry 211, 113014, 2021 | 14 | 2021 |
Targeting Non-Replicating Mycobacterium tuberculosis and Latent Infection: Alternatives and Perspectives (Mini-Review) A Egorova, EG Salina, V Makarov International Journal of Molecular Sciences 22 (24), 13317, 2021 | 13 | 2021 |
Nitric oxide-releasing compounds for the treatment of lung infections LR Chiarelli, G Degiacomi, A Egorova, V Makarov, MR Pasca Drug Discovery Today 26 (2), 542-550, 2021 | 10 | 2021 |
Design and Synthesis of Pyrano[3,2-b]indolones Showing Antimycobacterial Activity N Monakhova, J Korduláková, A Vocat, A Egorova, A Lepioshkin, ... ACS Infectious Diseases 7 (1), 88-100, 2020 | 8 | 2020 |
WIN compounds: on the way to efficient antipicornaviral agent. A historical survey AP Egorova, VA Makarov Russian Chemical Bulletin 69 (4), 635-646, 2020 | 7 | 2020 |
The Evolution of Pleconaril: Modified O-Alkyl Linker Analogs Have Biological Activity towards Coxsackievirus B3 Nancy A Volobueva, A Egorova, A Galochkina, S Ekins, V Zarubaev, V Makarov Molecules 25 (6), 1345, 2020 | 7 | 2020 |
Broad-spectrum antiviral diazadispiroalkane core molecules block attachment and cell-to-cell spread of herpesviruses A Dohme, M Knoblauch, A Egorova, V Makarov, E Bogner Antiviral Research 206, 105402, 2022 | 5 | 2022 |
A proof-of-concept study for the efficacy of dispirotripiperazine PDSTP in a rabbit model of herpes simplex epithelial keratitis L Alimbarova, A Egorova, O Riabova, N Monakhova, V Makarov Antiviral Research 202, 105327, 2022 | 4 | 2022 |
Efficacy of an isoxazole-3-carboxamide analog of pleconaril in mouse models of Enterovirus-D68 and Coxsackie B5 TR Lane, J Fu, B Sherry, B Tarbet, BL Hurst, O Riabova, E Kazakova, ... Antiviral Research 216, 105654, 2023 | 1 | 2023 |
Thienopyrimidines kill Mycobacterium tuberculosis by production of nitric oxide EG Salina, AP Egorova, LR Chiarelli, MR Pasca, VA Makarov FEBS Open Bio 8, 239-240, 2018 | 1 | 2018 |
Molecular mechanism of rhinovirus escape from the Pyrazolo [3, 4-d] pyrimidine capsid-binding inhibitor OBR-5-340 via mutations distant from the binding pocket: Derivatives … M Richter, K Döring, D Blaas, O Riabova, M Khrenova, E Kazakova, ... Antiviral Research 222, 105810, 2024 | | 2024 |
Antidepressant-like Effect of the Eburnamine-Type Molecule Vindeburnol in Rat and Mouse Models of Ultrasound-Induced Depression E Zubkov, O Riabova, Y Zorkina, A Egorova, V Ushakova, A Lepioshkin, ... ACS Chemical Neuroscience 15 (3), 560-571, 2024 | | 2024 |
SCRAPPY-a single cell rapid assay of proteome perturbation in yeast uncovers a joint role of aromatic amino acids and oxidative stress in the toxicity of lipophilic nucleoside … E Ghazy, VA Bidiuk, F Ryabov, OV Mitkevich, O Riabova, ... bioRxiv, 2024.02. 19.580949, 2024 | | 2024 |
Pyrrolo [2, 3-e] indazole as a novel chemotype for both influenza A virus and pneumococcal neuraminidase inhibitors A Egorova, M Richter, M Khrenova, E Dietrich, A Tsedilin, E Kazakova, ... RSC advances 13 (27), 18253-18261, 2023 | | 2023 |
Thieno[2,3‐d]pyrimidine‐Core Compounds Show Activity against Clinically Relevant Gram‐Positive Bacteria O Riabova, A Egorova, A Lepioshkin, Y Li, K Voigt, F Kloss, V Makarov ChemMedChem 17 (17), e202200207, 2022 | | 2022 |